effect of glutamate antagonist on pt with acute cerebral infarction = targets NMDA receptor
decreases calcium entry into neurons = decreased excitotoxicity = promotes recovery from acute cerebral infarction.
Tgouh nuieqt.os
aeclRl atth aeMimnent (hzal'msreie )ugdr si a NMAD eceRoptr soingtnAat tath slhep petvrne xxtyoiitcetco yb ikgonclB Ca+2 yetrn. ah'tsT hwo I errembem sih.t
a picture for better understanding https://2e.mindsmachine.com/asf04.02.html
^ link is dead :( (they published a 3/e) but here is the re-route to the new site if anyone wants to dig in https://learninglink.oup.com/access/watson3e-student-resources
MDNA rtsrepeco ni sith aecs era bigen dues rfo nglo rtme pineattntooi niitwh het raibn dna uot of all fo reteh ceoshci lnoy ihst rpceerto sseu C+a
I ekipdc NADM eubscae ’sti ruiya,ltstom tbu si rhete yan depeer asrone orf hst?i
You can rnwsae by psrosce fo nmoeaiinti.l t"pietmoievC tasinnieo"tcr ekmas uoy ntihk mtryaouitsl .TN ssCro out BAGA and ely.cing nI eth trexoc so at.ategulm poitobatcMre lduwo eamn ese'hrt ocsned seeenrssgm envdivlo adn the protcree owldu tno ttnrimsa muliac.c nceHe ANM.D
usde ni ongl ertm tinepttoiona ,ae(gaulng rmoy,)me yaM lsao alpy a oler in egne inprsantocirt in ronuesn
)1 NDMA si a aGulattme roertpce ytsu2b)pe PAAM is a tyusbep fo MDNA that is yalliniti iveattcad by gmtuatlea )3reelaes DAMN rerocetsp are duonf arne AMPA etsrcorpe utb ear ton aaetcitdv by wlo eselvl fo tlaaeugmt eesrael due ot a Mg oin ock’‘iglnb eht )4nn lecah etqneFur tAicon aloptenit g;—&t usimitonlat fo AMAP >— aospzdeielr psot anysictp ueonnr &g;t— eaoltgv eeenntpdd Mg bcklo of NAMD prterceo mdvoere 5) xulinf of aC tghohur DNAM ;—> eucsas even rmoe MAAP peesctror ot be eerditsn into teh rbaememn T(O:EN AMAP is resisneovp to Ca dan am u6g)aett)l aeueBsc eethr are emro etsrrcope to ndseorp to ,ti hte elcl is omer epvsisneor ot eautmtlga
lla hte hsreot a inpvteoitconem eicns hety ehva citcifecsicipieys(fp adsni,gl) MDAN is eht lyon nonccviheneees(elt mvopetticei r,)ptreceo ash a dlgain tsei dan ca , an dna gc.heemn.. tiepciomvte
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yM iamn kwa-Gealtae:stauya tm = rmajo yrcioxtaet t.etmteiorsarnnur Tow tepys fo p)cror1:se te oopc,abimettr stom of ihcwh era rptscypnaei Gi hwihc adels ot ddecaeres MAND oecreptr cvayitit dna rsik fo iyticixixoco,tet or cysitostnpap Gq rpeeorsct thta dela ot secranei Na+, ,+K dna dceerades etulagtma uasces depnoaotalzrii nad sdraceine +g+M esdetcminpla nad MADN roeprcte tvyactii dna rski fo yxcoc,itxietoti nad ) 2 ocinooptri nalcnshe lgudniicn ADMN dan k/eaMinPAAta ,ecnslnha iwhhc all lwoal fceipcsonin iotnca ufxi,ln utb nlyo ANDM lwlaso C++a ilufxn (and oyln ni a leoavgt peeendtnd mneran aetrf stenffiicu eaptidnozarlio sah eicasldpd teh othbniiri +M+g ion ni eth ean)c.lhn
BAGA dna ylniegc = nbtoiirihy eruneitr.sstramotn 1) GAAB-A dan G-AACB = itncriooop aenclsnh htta aeld ot lexfu fo ,C-l dna tiepesd ihts ugacnis aznieporatdi,ol eht unnero itlsl ssayt owelb rgetnsi atnleio.pt A-GAAB dibnign tsei for trtuabse,abir ,tiseodrs GAAB, nda tiroocnipx = niesdi opre of hnncea.l B-AAGA nigdinb itse of pezseideozabinn = iseudot of rpeo fo nhaecl.n )2 lcGiney cnehanl si a yevr alirsmi -lC elxfu .haecnnl 3 ) ABG-AB is a btaroocpmeti anhencl taht iatsactev iG lngiade to rddacseee cAPM hwhci eivtaatcs fuexfl +K nacehlsn nda sbniitih +Ca+ filunx enhncasl iadlgen ot hriorniotplzae.ayp
oeBcngii aenmis = ctmiaaleesnhoc eanpmdoi oitcodroinna( fo bydo tvo,nmeme earr,wd aviion,tmot )neocrtifren,em rpepnernenhioi ee(lps, nlkfs,sewaue non,tettai fiegend e,rhoiabv rnpeheneipi lewsot( cncraoonittne in CS,)N lusp rsoteinno le,(pse nklfwseause, eoeirdnps,s aeiytn,x a)euasn nda ienahismt a(ru,aols ett,ianton g,llerya tiusse g,mdeaa and aym nnicuefle lobdo riabn )fl.ow ublO,iysov lal of isth si in dodaitin ot gicrdaenre rnnoreassmiositun and ,flihgt ,tgrhif adn ghtif neseorp.s
ATP nda rheot isurenp = ctrytaioxe s,ssominairnt cerol-eaesd thiw hoert easmll-uolceml tse.toeurrsntarimn enndosieA n'tsi lsclicalays dreednosci a erorrtnastnemuti acuesbe it st'in asdd/erstloeree in +C+a denndetep anmn,re tbu evdredi romf APT ofereb ngiahv na ttciyraoex lpn.etatoi
otcehlylnieAc = ojamr timnrrntetaoesru nlodeivv ni isrsntnsmeanoiruo via smcruina dna coitininc rpsoee.rtc
ePipted teatmristnernuors = cmlyoomn eeralesd sa eprpodietp argerl esoruscrpr htta are ceavled by fieispcc yezmens htta were in eht sema snrttnoremreiatu selevci unop sarl.eee iveF ypste = rainbg/ut p,sdtieep doipio pdt,piese rpyiutati t,ipspde cyaahihtpmol lnieserga ,rnomhseo nda osteh not lsca.siiedf elpaExms = ruocerspr atth sevgi isre to stbunasce P oi(ucpaphsp,m ,xoenrocet nda TIG nda deleersa form llmas mirteaed NPS C ifsrbe taht atmistrn pnia nda reeamuteptr innriomato,f leouwpfr hyspoievetn, dnteihibi by podiio sdp)eptie, ineuioknrn A, dpopeitunere ,K dna uepoetpnedri ,gamam nda piodio deseppit igcunnidl pntal sialdokla ei(kl omr,iehnp) sttyinhce ipdooi aie,vdrvesit nad nrnpdsio,he hyspd,irnno and pheasil.nkne nI galnree podiio iesdptpe aer ntssspderea i..(e lasgeaian nmmeaih,sc) vnvileod in loecxmp irbehsoav l(uaexs ta,toatirnc erisvaesibvguis/esmgs )hoaevb,irs nda alempdicti (uhgoht otn neditvfi)ei ni siytrcpahic srdo.ersid
llre,aOv tintssarreeurnmto = ypte sptey: oul-cllmlamees msaerrtttisn dna onuepited,sper erewh caeomlulls-lmes ttmesartsinr era fretsa and etaeimd iadrp taspiycn trinimsonssa ei.(. orndneag SNS /fhitg/lfgihrtgihft icukq rsosep)e,n wheer as eednopreutpsi (gnaol tiwh oglciibo sinmae adn omse amlsl ceolmleu sitant)tsrmre rea erwosl and maedeti laarg,ud ndogpreol ii.rnnsssmunareoto
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